+Search query
-Structure paper
Title | The discovery of potent and selective pyridopyrimidin-7-one based inhibitors of B-Raf(V600E) kinase. |
---|---|
Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 22, Page 3387-3391, Year 2012 |
Publish date | Mar 13, 2012 (structure data deposition date) |
Authors | Ren, L. / Ahrendt, K.A. / Grina, J. / Laird, E.R. / Buckmelter, A.J. / Hansen, J.D. / Newhouse, B. / Moreno, D. / Wenglowsky, S. / Dinkel, V. ...Ren, L. / Ahrendt, K.A. / Grina, J. / Laird, E.R. / Buckmelter, A.J. / Hansen, J.D. / Newhouse, B. / Moreno, D. / Wenglowsky, S. / Dinkel, V. / Gloor, S.L. / Hastings, G. / Rana, S. / Rasor, K. / Risom, T. / Sturgis, H.L. / Voegtli, W.C. / Mathieu, S. |
External links | Bioorg. Med. Chem. Lett. / PubMed:22534450 |
Methods | X-ray diffraction |
Resolution | 3.6 Å |
Structure data | PDB-4e4x: |
Chemicals | ChemComp-T1Q: |
Source |
|
Keywords | Transferase/Transferase Inhibitor / Kinase / Transferase-Transferase Inhibitor complex |