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-Structure paper
Title | Multimode, cooperative mechanism of action of allosteric HIV-1 integrase inhibitors. |
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Journal, issue, pages | J. Biol. Chem., Vol. 287, Page 16801-16811, Year 2012 |
Publish date | Feb 8, 2012 (structure data deposition date) |
![]() | Kessl, J.J. / Jena, N. / Koh, Y. / Taskent-Sezgin, H. / Slaughter, A. / Feng, L. / de Silva, S. / Wu, L. / Le Grice, S.F. / Engelman, A. ...Kessl, J.J. / Jena, N. / Koh, Y. / Taskent-Sezgin, H. / Slaughter, A. / Feng, L. / de Silva, S. / Wu, L. / Le Grice, S.F. / Engelman, A. / Fuchs, J.R. / Kvaratskhelia, M. |
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Methods | X-ray diffraction |
Resolution | 2.45 Å |
Structure data | ![]() PDB-4dmn: |
Chemicals | ![]() ChemComp-ARS: ![]() ChemComp-SO4: ![]() ChemComp-0L9: ![]() ChemComp-HOH: |
Source |
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![]() | VIRAL PROTEIN/Inhibitor / Integrase / CCD / DDE motif / dimer interface / VIRAL PROTEIN-Inhibitor complex |