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-Structure paper
Title | Synthesis and Evaluation of Triazolones as Checkpoint Kinase 1 Inhibitors. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 22, Page 2330-, Year 2012 |
Publish date | Mar 30, 2011 (structure data deposition date) |
![]() | Oza, V. / Ashwell, S. / Brassil, P. / Breed, J. / Ezhuthachan, J. / Deng, C. / Grondine, M. / Horn, C. / Liu, D. / Lyne, P. ...Oza, V. / Ashwell, S. / Brassil, P. / Breed, J. / Ezhuthachan, J. / Deng, C. / Grondine, M. / Horn, C. / Liu, D. / Lyne, P. / Newcombe, N. / Pass, M. / Read, J. / Su, M. / Toader, D. / Yu, D. / Yu, Y. / Zabludoff, S. |
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Methods | X-ray diffraction |
Resolution | 1.3 - 1.83 Å |
Structure data | ![]() PDB-2yer: ![]() PDB-2yex: |
Chemicals | ![]() ChemComp-TQ1: ![]() ChemComp-SO4: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-GOL: ![]() ChemComp-YEX: |
Source |
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