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-Structure paper
Title | Structural basis of selective inhibition of human tankyrases. |
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Journal, issue, pages | J. Med. Chem., Vol. 55, Page 1360-1367, Year 2012 |
Publish date | Oct 19, 2011 (structure data deposition date) |
![]() | Narwal, M. / Venkannagari, H. / Lehtio, L. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.75 - 2.3 Å |
Structure data | ![]() PDB-3u9h: ![]() PDB-3u9y: ![]() PDB-3ua9: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-SO4: ![]() ChemComp-NCA: ![]() ChemComp-GOL: ![]() ChemComp-PEG: ![]() ChemComp-HOH: ![]() ChemComp-09L: ![]() ChemComp-IWR: |
Source |
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![]() | TRANSFERASE / PROTEIN-LIGAND COMPLEX / DIPHTHERIA TOXIN LIKE FOLD / ADP-RIBOSYLATION / TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE-TRANSFERASE INHIBITOR complex |