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-Structure paper
| Title | Identification of triazolopyridazinones as potent p38alpha inhibitors. |
|---|---|
| Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 22, Page 1226-1229, Year 2012 |
| Publish date | Oct 17, 2011 (structure data deposition date) |
Authors | Herberich, B. / Jackson, C. / Wurz, R.P. / Pettus, L.H. / Sherman, L. / Liu, Q. / Henkle, B. / Saris, C.J. / Wong, L.M. / Chmait, S. ...Herberich, B. / Jackson, C. / Wurz, R.P. / Pettus, L.H. / Sherman, L. / Liu, Q. / Henkle, B. / Saris, C.J. / Wong, L.M. / Chmait, S. / Lee, M.R. / Mohr, C. / Hsieh, F. / Tasker, A.S. |
External links | Bioorg. Med. Chem. Lett. / PubMed:22196117 |
| Methods | X-ray diffraction |
| Resolution | 2.15 Å |
| Structure data | ![]() PDB-3u8w: |
| Chemicals | ![]() ChemComp-09J: ![]() ChemComp-HOH: |
| Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / Serine/Threonine Protein Kinase / Transferase / TRANSFERASE-TRANSFERASE INHIBITOR complex |
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homo sapiens (human)
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