+Search query
-Structure paper
Title | Discovery of Novel, Potent, and Selective Inhibitors of 3-Phosphoinositide-Dependent Kinase (PDK1). |
---|---|
Journal, issue, pages | J. Med. Chem., Vol. 54, Page 8490-8500, Year 2011 |
Publish date | May 9, 2011 (structure data deposition date) |
Authors | Murphy, S.T. / Alton, G. / Bailey, S. / Baxi, S.M. / Burke, B.J. / Chappie, T.A. / Ermolieff, J. / Ferre, R. / Greasley, S. / Hickey, M. ...Murphy, S.T. / Alton, G. / Bailey, S. / Baxi, S.M. / Burke, B.J. / Chappie, T.A. / Ermolieff, J. / Ferre, R. / Greasley, S. / Hickey, M. / Humphrey, J. / Kablaoui, N. / Kath, J. / Kazmirski, S. / Kraus, M. / Kupchinsky, S. / Li, J. / Lingardo, L. / Marx, M.A. / Richter, D. / Tanis, S.P. / Tran, K. / Vernier, W. / Xie, Z. / Yin, M.J. / Yu, X.H. |
External links | J. Med. Chem. / PubMed:22040023 |
Methods | X-ray diffraction |
Resolution | 1.92 - 2.55 Å |
Structure data | PDB-3rwp: PDB-3rwq: |
Chemicals | ChemComp-GOL: ChemComp-SO4: ChemComp-ABQ: ChemComp-HOH: ChemComp-3RW: |
Source |
|
Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / Kinase domain / Transferase / Phosphoserine: SEP / TRANSFERASE-TRANSFERASE INHIBITOR complex |