+Search query
-Structure paper
Title | Novel isoquinolone PDK1 inhibitors discovered through fragment-based lead discovery. |
---|---|
Journal, issue, pages | J Comput Aided Mol Des, Vol. 25, Page 689-698, Year 2011 |
Publish date | Jun 6, 2011 (structure data deposition date) |
![]() | Johnson, M.C. / Hu, Q. / Lingardo, L. / Ferre, R.A. / Greasley, S. / Yan, J. / Kath, J. / Chen, P. / Ermolieff, J. / Alton, G. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.7 Å |
Structure data | ![]() PDB-3sc1: |
Chemicals | ![]() ChemComp-3S1: ![]() ChemComp-SO4: ![]() ChemComp-GOL: ![]() ChemComp-HOH: |
Source |
|
![]() | TRANSFERASE/TRANSFERASE INHIBITOR / KINASE DOMAIN / PHOSPHOSERINE / SEP / TRANSFERASE-TRANSFERASE INHIBITOR complex |