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-Structure paper
Title | Small Molecule Agonists of the Orphan Nuclear Receptors Steroidogenic Factor-1 (SF-1, NR5A1) and Liver Receptor Homologue-1 (LRH-1, NR5A2). |
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Journal, issue, pages | J. Med. Chem., Vol. 54, Page 2266-2281, Year 2011 |
Publish date | Nov 15, 2010 (structure data deposition date) |
![]() | Whitby, R.J. / Stec, J. / Blind, R.D. / Dixon, S. / Leesnitzer, L.M. / Orband-Miller, L.A. / Williams, S.P. / Willson, T.M. / Xu, R. / Zuercher, W.J. ...Whitby, R.J. / Stec, J. / Blind, R.D. / Dixon, S. / Leesnitzer, L.M. / Orband-Miller, L.A. / Williams, S.P. / Willson, T.M. / Xu, R. / Zuercher, W.J. / Cai, F. / Ingraham, H.A. |
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Methods | X-ray diffraction |
Resolution | 1.75 Å |
Structure data | ![]() PDB-3plz: |
Chemicals | ![]() ChemComp-470: ![]() ChemComp-EDO: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION/RECEPTOR/AGONIST / alpha helical sandwhich / nuclear receptor / family five / transcription factor / co-activator / TRANSCRIPTION-RECEPTOR-AGONIST complex |