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Title5-Amino-pyrazoles as potent and selective p38α inhibitors
Journal, issue, pagesBioorg. Med. Chem. Lett., Vol. 20, Page 6886-6889, Year 2010
Publish dateAug 10, 2010 (structure data deposition date)
AuthorsDas, J. / Moquin, R.V. / Dyckman, A.J. / Li, T. / Pitt, S. / Zhang, R. / Shen, D.R. / McIntyre, K.W. / Gillooly, K. / Doweyko, A.M. ...Das, J. / Moquin, R.V. / Dyckman, A.J. / Li, T. / Pitt, S. / Zhang, R. / Shen, D.R. / McIntyre, K.W. / Gillooly, K. / Doweyko, A.M. / Newitt, J.A. / Sack, J.S. / Zhang, H. / Kiefer, S.E. / Kish, K. / McKinnon, M. / Barrish, J.C. / Dodd, J.H. / Schieven, G.L. / Leftheris, K.
External linksBioorg. Med. Chem. Lett. / PubMed:21035336
MethodsX-ray diffraction
Resolution2.21 Å
Structure data

PDB-3ocg:
P38 Alpha kinase complexed with a 5-amino-pyrazole based inhibitor
Method: X-RAY DIFFRACTION / Resolution: 2.21 Å

Chemicals

ChemComp-OCG:
5-amino-N-[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]-1-phenyl-1H-pyrazole-4-carboxamide

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsTRANSFERASE/TRANSFERASE INHIBITOR / P38 map kinase / serine/threonine-protein kinase / transferase / TRANSFERASE-TRANSFERASE INHIBITOR complex

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