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-Structure paper
Title | Structure-based approach to nanomolar, water soluble matrix metalloproteinases inhibitors (MMPIs). |
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Journal, issue, pages | Eur. J. Med. Chem., Vol. 45, Page 5919-5925, Year 2010 |
Publish date | May 19, 2010 (structure data deposition date) |
Authors | Attolino, E. / Calderone, V. / Dragoni, E. / Fragai, M. / Richichi, B. / Luchinat, C. / Nativi, C. |
External links | Eur. J. Med. Chem. / PubMed:20965620 |
Methods | X-ray diffraction |
Resolution | 1.55 - 1.81 Å |
Structure data | PDB-3n2u: PDB-3n2v: |
Chemicals | ChemComp-ZN: ChemComp-CA: ChemComp-D3X: ChemComp-HOH: ChemComp-JT5: |
Source |
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Keywords | Hydrolase/Hydrolase inhibitor / MATRIX METALLOPROTEINASE / MMP12 / ELASTASE / COMPLEX (ELASTASE-INHIBITOR) / METALLO ELASTASE / EXTRACELLULAR MATRIX / GLYCOPROTEIN / HYDROLASE / METAL-INDING / METALLOPROTEASE / PROTEASE / SECRETED / ZYMOGEN / Hydrolase-Hydrolase inhibitor complex |