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-Structure paper
Title | Design, Synthesis and Evaluation of Indolinones as Inhibitors of the Transforming Growth Factor Beta Receptor I (Tgfbri) |
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Journal, issue, pages | J. Med. Chem., Vol. 53, Page 7287-, Year 2010 |
Publish date | Mar 3, 2010 (structure data deposition date) |
Authors | Roth, G.J. / Heckel, A. / Brandl, T. / Grauert, M. / Hoerer, S. / Kley, J.T. / Schnapp, G. / Baum, P. / Mennerich, D. / Schnapp, A. / Park, J.E. |
External links | J. Med. Chem. / PubMed:20919678 |
Methods | X-ray diffraction |
Resolution | 3.7 Å |
Structure data | PDB-2x7o: |
Chemicals | ChemComp-ZOP: |
Source |
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Keywords | TRANSFERASE / KINASE / GLYCOPROTEIN |