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-Structure paper
Title | A novel series of positive modulators of the AMPA receptor: discovery and structure based hit-to-lead studies. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 20, Page 5753-5756, Year 2010 |
Publish date | Jul 22, 2010 (structure data deposition date) |
![]() | Jamieson, C. / Basten, S. / Campbell, R.A. / Cumming, I.A. / Gillen, K.J. / Gillespie, J. / Kazemier, B. / Kiczun, M. / Lamont, Y. / Lyons, A.J. ...Jamieson, C. / Basten, S. / Campbell, R.A. / Cumming, I.A. / Gillen, K.J. / Gillespie, J. / Kazemier, B. / Kiczun, M. / Lamont, Y. / Lyons, A.J. / Maclean, J.K. / Moir, E.M. / Morrow, J.A. / Papakosta, M. / Rankovic, Z. / Smith, L. |
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Methods | X-ray diffraction |
Resolution | 1.9 - 2.02 Å |
Structure data | ![]() PDB-3o28: ![]() PDB-3o29: ![]() PDB-3o2a: |
Chemicals | ![]() ChemComp-O28: ![]() ChemComp-GLU: ![]() ChemComp-SO4: ![]() ChemComp-DMS: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-O29: ![]() ChemComp-O30: |
Source |
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![]() | TRANSPORT PROTEIN / Membrane Protein / Fusion protein / chimera protein |