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-Structure paper
Title | Application of Chemoproteomics to Drug Discovery: Identification of a Clinical Candidate Targeting Hsp90. |
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Journal, issue, pages | Chem. Biol., Vol. 17, Page 686-694, Year 2010 |
Publish date | Apr 22, 2010 (structure data deposition date) |
Authors | Fadden, P. / Huang, K.H. / Veal, J.M. / Steed, P.M. / Barabasz, A.F. / Foley, B. / Hu, M. / Partridge, J.M. / Rice, J. / Scott, A. ...Fadden, P. / Huang, K.H. / Veal, J.M. / Steed, P.M. / Barabasz, A.F. / Foley, B. / Hu, M. / Partridge, J.M. / Rice, J. / Scott, A. / Dubois, L.G. / Freed, T.A. / Silinski, M.A. / Barta, T.E. / Hughes, P.F. / Ommen, A. / Ma, W. / Smith, E.D. / Spangenberg, A.W. / Eaves, J. / Hanson, G.J. / Hinkley, L. / Jenks, M. / Lewis, M. / Otto, J. / Pronk, G.J. / Verleysen, K. / Haystead, T.A. / Hall, S.E. |
External links | Chem. Biol. / PubMed:20659681 |
Methods | X-ray diffraction |
Resolution | 1.9 Å |
Structure data | PDB-3mnr: |
Chemicals | ChemComp-SD1: ChemComp-HOH: |
Source |
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Keywords | CHAPERONE / HSP90 / HEAT SHOCK PROTEIN 90 / PROTEIN-LIGAND COMPLEX |