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-Structure paper
Title | Crystal Structures of HIV-1 Reverse Transcriptase with Etravirine (TMC125) and Rilpivirine (TMC278): Implications for Drug Design. |
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Journal, issue, pages | J. Med. Chem., Vol. 53, Page 4295-4299, Year 2010 |
Publish date | Mar 31, 2010 (structure data deposition date) |
Authors | Lansdon, E.B. / Brendza, K.M. / Hung, M. / Wang, R. / Mukund, S. / Jin, D. / Birkus, G. / Kutty, N. / Liu, X. |
External links | J. Med. Chem. / PubMed:20438081 |
Methods | X-ray diffraction |
Resolution | 2.3 - 2.8 Å |
Structure data | PDB-3mec: PDB-3med: PDB-3mee: PDB-3meg: |
Chemicals | ChemComp-65B: ChemComp-SO4: ChemComp-HOH: ChemComp-CL: ChemComp-T27: |
Source |
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Keywords | TRANSFERASE / HIV / reverse transcriptase / TMC125 / etravirine / NNRTI / TMC278 / rilpivirine |