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| Title | Targeting Bcr-Abl by combining allosteric with ATP-binding-site inhibitors. |
|---|---|
| Journal, issue, pages | Nature, Vol. 463, Page 501-506, Year 2010 |
| Publish date | Oct 8, 2009 (structure data deposition date) |
Authors | Zhang, J. / Adrian, F.J. / Jahnke, W. / Cowan-Jacob, S.W. / Li, A.G. / Iacob, R.E. / Sim, T. / Powers, J. / Dierks, C. / Sun, F. ...Zhang, J. / Adrian, F.J. / Jahnke, W. / Cowan-Jacob, S.W. / Li, A.G. / Iacob, R.E. / Sim, T. / Powers, J. / Dierks, C. / Sun, F. / Guo, G.R. / Ding, Q. / Okram, B. / Choi, Y. / Wojciechowski, A. / Deng, X. / Liu, G. / Fendrich, G. / Strauss, A. / Vajpai, N. / Grzesiek, S. / Tuntland, T. / Liu, Y. / Bursulaya, B. / Azam, M. / Manley, P.W. / Engen, J.R. / Daley, G.Q. / Warmuth, M. / Gray, N.S. |
External links | Nature / PubMed:20072125 |
| Methods | X-ray diffraction |
| Resolution | 1.74 Å |
| Structure data | ![]() PDB-3k5v: |
| Chemicals | ![]() ChemComp-STJ: ![]() ChemComp-STI: ![]() ChemComp-CL: ![]() ChemComp-HOH: |
| Source |
|
Keywords | TRANSFERASE / kinase / ATP-binding / Nucleotide-binding / Oncogene / SH2 domain / Tyrosine-protein kinase |
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