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-Structure paper
| Title | Discovery of C-imidazole azaheptapyridine FPT inhibitors. |
|---|---|
| Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 20, Page 1134-1136, Year 2010 |
| Publish date | Nov 23, 2009 (structure data deposition date) |
Authors | Zhu, H.Y. / Cooper, A.B. / Desai, J. / Njoroge, G. / Kirschmeier, P. / Bishop, W.R. / Strickland, C. / Hruza, A. / Doll, R.J. / Girijavallabhan, V.M. |
External links | Bioorg. Med. Chem. Lett. / PubMed:20056542 |
| Methods | X-ray diffraction |
| Resolution | 2.1 Å |
| Structure data | ![]() PDB-3ksq: |
| Chemicals | ![]() ChemComp-MG: ![]() ChemComp-ZN: ![]() ChemComp-FPP: ![]() ChemComp-Z96: ![]() ChemComp-HOH: |
| Source |
|
Keywords | TRANSFERASE / PRENYLTRANSFERASE / Metal-binding / Phosphoprotein |
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