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TitleBioisosterism of urea-based GCPII inhibitors: Synthesis and structure-activity relationship studies.
Journal, issue, pagesBioorg. Med. Chem. Lett., Vol. 20, Page 392-397, Year 2010
Publish dateSep 3, 2009 (structure data deposition date)
AuthorsWang, H. / Byun, Y. / Barinka, C. / Pullambhatla, M. / Bhang, H.E. / Fox, J.J. / Lubkowski, J. / Mease, R.C. / Pomper, M.G.
External linksBioorg. Med. Chem. Lett. / PubMed:19897367
MethodsX-ray diffraction
Resolution2.3 Å
Structure data

PDB-3iww:
Crystal structure of human glutamate carboxypeptidase II (GCPII) in a complex with DBIBzL, a urea-based inhibitor
Method: X-RAY DIFFRACTION / Resolution: 2.3 Å

Chemicals

ChemComp-ZN:
Unknown entry

ChemComp-CA:
Unknown entry

ChemComp-CL:
Unknown entry

ChemComp-NAG:
2-acetamido-2-deoxy-beta-D-glucopyranose

ChemComp-YZE:
N~2~-{[(1S)-1-carboxybut-3-en-1-yl]carbamoyl}-N~6~-[(4-iodophenyl)carbonyl]-L-lysine

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsHYDROLASE / prostate specific membrane antigen; metallopeptidase; folate hydrolase; glutamate carboxypeptidase II; Naaladase; urea-based inhibitor / Carboxypeptidase / Cell membrane / Dipeptidase / Glycoprotein / Membrane / Metal-binding / Metalloprotease / Multifunctional enzyme / Protease / Signal-anchor / Transmembrane

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