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-Structure paper
Title | Inhibition of tumor cell growth, invasion, and metastasis by EXEL-2880 (XL880, GSK1363089), a novel inhibitor of HGF and VEGF receptor tyrosine kinases. |
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Journal, issue, pages | Cancer Res., Vol. 69, Page 8009-8016, Year 2009 |
Publish date | Feb 8, 2010 (structure data deposition date) |
Authors | Qian, F. / Engst, S. / Yamaguchi, K. / Yu, P. / Won, K.A. / Mock, L. / Lou, T. / Tan, J. / Li, C. / Tam, D. ...Qian, F. / Engst, S. / Yamaguchi, K. / Yu, P. / Won, K.A. / Mock, L. / Lou, T. / Tan, J. / Li, C. / Tam, D. / Lougheed, J. / Yakes, F.M. / Bentzien, F. / Xu, W. / Zaks, T. / Wooster, R. / Greshock, J. / Joly, A.H. |
External links | Cancer Res. / PubMed:19808973 |
Methods | X-ray diffraction |
Resolution | 2.02 Å |
Structure data | PDB-3lq8: |
Chemicals | ChemComp-88Z: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / kinase domain / XL880 / GSK1363089 / ATP-binding / Kinase / Nucleotide-binding / Phosphoprotein / Proto-oncogene / Receptor / Transmembrane / Tyrosine-protein kinase |