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-Structure paper
Title | Inhibitors selective for mycobacterial versus human proteasomes. |
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Journal, issue, pages | Nature, Vol. 461, Page 621-626, Year 2009 |
Publish date | Apr 23, 2009 (structure data deposition date) |
![]() | Lin, G. / Li, D. / de Carvalho, L.P. / Deng, H. / Tao, H. / Vogt, G. / Wu, K. / Schneider, J. / Chidawanyika, T. / Warren, J.D. ...Lin, G. / Li, D. / de Carvalho, L.P. / Deng, H. / Tao, H. / Vogt, G. / Wu, K. / Schneider, J. / Chidawanyika, T. / Warren, J.D. / Li, H. / Nathan, C. |
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Methods | X-ray diffraction |
Resolution | 2.43 - 2.878 Å |
Structure data | ![]() PDB-3h6f: ![]() PDB-3h6i: ![]() PDB-3hf9: ![]() PDB-3hfa: |
Chemicals | ![]() ChemComp-DMF: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE / Binding Sites / Oxazolidin-2-one / Mycobacterium tuberculosis / Protease Inhibitors / Proteasome Endopeptidase Complex / Protein Subunits / Substrate Specificity / Proteasome / open gate / mutant / Proteasome Endopeptidase |