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-Structure paper
Title | Identification of PDE4B Over 4D subtype-selective inhibitors revealing an unprecedented binding mode |
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Journal, issue, pages | Bioorg. Med. Chem., Vol. 17, Page 5336-5341, Year 2009 |
Publish date | May 29, 2009 (structure data deposition date) |
Authors | Kranz, M. / Wall, M. / Evans, B. / Miah, A. / Ballantine, S. / Delves, C. / Dombroski, B. / Gross, J. / Schneck, J. / Villa, J.P. ...Kranz, M. / Wall, M. / Evans, B. / Miah, A. / Ballantine, S. / Delves, C. / Dombroski, B. / Gross, J. / Schneck, J. / Villa, J.P. / Neu, M. / Somers, D.O. |
External links | Bioorg. Med. Chem. / PubMed:19525117 |
Methods | X-ray diffraction |
Resolution | 2.23 Å |
Structure data | PDB-3hmv: |
Chemicals | ChemComp-ZN: ChemComp-MG: ChemComp-HBT: ChemComp-GOL: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / PDE / PHOSPHODIESTERASE / cAMP / Alternative splicing / Phosphoprotein / Polymorphism |