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-Structure paper
| Title | Discovery and Characterization of a Highly Selective Faah Inhibitor that Reduces Inflammatory Pain. |
|---|---|
| Journal, issue, pages | Chem. Biol., Vol. 16, Page 411-, Year 2009 |
| Publish date | Feb 11, 2009 (structure data deposition date) |
Authors | Ahn, K. / Johnson, D.S. / Mileni, M. / Beidler, D. / Long, J.Z. / Mckinney, M.K. / Weerapana, E. / Sadagopan, N. / Liimatta, M. / Smith, S.E. ...Ahn, K. / Johnson, D.S. / Mileni, M. / Beidler, D. / Long, J.Z. / Mckinney, M.K. / Weerapana, E. / Sadagopan, N. / Liimatta, M. / Smith, S.E. / Lazerwith, S. / Stiff, C. / Kamtekar, S. / Bhattacharya, K. / Zhang, Y. / Swaney, S. / Vanbecelaere, K. / Stevens, R.C. / Cravatt, B.F. |
External links | Chem. Biol. / PubMed:19389627 |
| Methods | X-ray diffraction |
| Resolution | 2.8 Å |
| Structure data | ![]() PDB-2wap: |
| Chemicals | ![]() ChemComp-PIX: ![]() ChemComp-CL: ![]() ChemComp-NA: ![]() ChemComp-HOH: |
| Source |
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Keywords | HYDROLASE / FATTY ACID AMIDE HYDROLASE / UREA INHIBITOR / GOLGI APPARATUS / ENDOPLASMIC RETICULUM / ACYL- ENZYME / TRANSMEMBRANE / PHOSPHOPROTEIN / FAAH / DRUG / MEMBRANE / INHIBITOR |
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