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-Structure paper
Title | Structural basis for inhibitor specificity in human poly(ADP-ribose) polymerase-3. |
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Journal, issue, pages | J. Med. Chem., Vol. 52, Page 3108-3111, Year 2009 |
Publish date | Jan 29, 2008 (structure data deposition date) |
Authors | Lehtio, L. / Jemth, A.S. / Collins, R. / Loseva, O. / Johansson, A. / Markova, N. / Hammarstrom, M. / Flores, A. / Holmberg-Schiavone, L. / Weigelt, J. ...Lehtio, L. / Jemth, A.S. / Collins, R. / Loseva, O. / Johansson, A. / Markova, N. / Hammarstrom, M. / Flores, A. / Holmberg-Schiavone, L. / Weigelt, J. / Helleday, T. / Schuler, H. / Karlberg, T. |
External links | J. Med. Chem. / PubMed:19354255 |
Methods | X-ray diffraction |
Resolution | 2.1 - 2.8 Å |
Structure data | PDB-3c49: PDB-3c4h: PDB-3ce0: PDB-3fhb: |
Chemicals | ChemComp-KU8: ChemComp-HOH: ChemComp-DRL: ChemComp-DMS: ChemComp-P34: ChemComp-GAB: |
Source |
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Keywords | TRANSFERASE / enzyme-inhibitor complex / catalytic fragment / Structural Genomics / Structural Genomics Consortium / SGC / Alternative splicing / Glycosyltransferase / NAD / Nucleus |