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-Structure paper
Title | Fragment-based Identification of Hsp90 Inhibitors. |
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Journal, issue, pages | Chemmedchem, Vol. 4, Page 963-966, Year 2009 |
Publish date | Jan 12, 2009 (structure data deposition date) |
Authors | Barker, J.J. / Barker, O. / Boggio, R. / Chauhan, V. / Cheng, R.K. / Corden, V. / Courtney, S.M. / Edwards, N. / Falque, V.M. / Fusar, F. ...Barker, J.J. / Barker, O. / Boggio, R. / Chauhan, V. / Cheng, R.K. / Corden, V. / Courtney, S.M. / Edwards, N. / Falque, V.M. / Fusar, F. / Gardiner, M. / Hamelin, E.M. / Hesterkamp, T. / Ichihara, O. / Jones, R.S. / Mather, O. / Mercurio, C. / Minucci, S. / Montalbetti, C.A. / Muller, A. / Patel, D. / Phillips, B.G. / Varasi, M. / Whittaker, M. / Winkler, D. / Yarnold, C.J. |
External links | Chemmedchem / PubMed:19301319 |
Methods | X-ray diffraction |
Resolution | 1.9 - 2 Å |
Structure data | PDB-3ft5: PDB-3ft8: |
Chemicals | ChemComp-MO8: ChemComp-HOH: ChemComp-MOJ: |
Source |
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Keywords | CHAPERONE / HSP90 N-terminal nucleotide binding domain / Alternative splicing / ATP-binding / Cytoplasm / Nucleotide-binding / Phosphoprotein / Stress response |