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TitleStructural analysis of ARC-type inhibitor (ARC-1034) binding to protein kinase A catalytic subunit and rational design of bisubstrate analogue inhibitors of basophilic protein kinases.
Journal, issue, pagesJ. Med. Chem., Vol. 52, Page 308-321, Year 2009
Publish dateJan 9, 2008 (structure data deposition date)
AuthorsLavogina, D. / Lust, M. / Viil, I. / Konig, N. / Raidaru, G. / Rogozina, J. / Enkvist, E. / Uri, A. / Bossemeyer, D.
External linksJ. Med. Chem. / PubMed:19143565
MethodsX-ray diffraction
Resolution2.3 Å
Structure data

PDB-3bwj:
Complex of PKA with the bisubstrate protein kinase inhibitor lead compound Arc-1034
Method: X-RAY DIFFRACTION / Resolution: 2.3 Å

Chemicals

ChemComp-ARX:
(2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-(6-{[(1R)-4-carbamimidamido-1-{[(1R)-4-carbamimidamido-1-carbamoylbutyl]carbamoyl}butyl]amino}-6-oxohexyl)-3,4-dihydroxytetrahydrofuran-2-carboxamide

ChemComp-HOH:
WATER

Source
  • bos taurus (domestic cattle)
KeywordsTRANSFERASE/TRANSFERASE INHIBITOR / bisubstrate inhibitor / protein kinase / Serine/threonine-protein kinase / ATP-binding / cAMP / Phosphoprotein / TRANSFERASE-TRANSFERASE INHIBITOR complex

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