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-Structure paper
Title | Optimizing Natural Products by Biosynthetic Engineering: Discovery of Nonquinone Hsp90 Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 51, Page 5494-, Year 2008 |
Publish date | Jun 16, 2008 (structure data deposition date) |
Authors | Zhang, M.Q. / Gaisser, S. / Nur-E-Alam, M. / Sheehan, L.S. / Vousden, W.A. / Gaitatzis, N. / Peck, G. / Coates, N.J. / Moss, S.J. / Radzom, M. ...Zhang, M.Q. / Gaisser, S. / Nur-E-Alam, M. / Sheehan, L.S. / Vousden, W.A. / Gaitatzis, N. / Peck, G. / Coates, N.J. / Moss, S.J. / Radzom, M. / Foster, T.A. / Sheridan, R.M. / Gregory, M.A. / Roe, S.M. / Prodromou, C. / Pearl, L.H. / Boyd, S.M. / Wilkinson, B. / Martin, C.J. |
External links | J. Med. Chem. / PubMed:18800759 |
Methods | X-ray diffraction |
Resolution | 1.9 Å |
Structure data | PDB-2vw5: |
Chemicals | ChemComp-BC6: ChemComp-SO4: ChemComp-HOH: |
Source |
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Keywords | CHAPERONE / ATPASE / CYTOPLASM / INHIBITOR / ATP-BINDING / STRESS RESPONSE / NUCLEOTIDE-BINDING |