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-Structure paper
Title | Discovery of a novel class of PPARdelta partial agonists |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 18, Page 5018-5022, Year 2008 |
Publish date | Jul 25, 2008 (structure data deposition date) |
Authors | Shearer, B.G. / Patel, H.S. / Billin, A.N. / Way, J.M. / Winegar, D.A. / Lambert, M.H. / Xu, R.X. / Leesnitzer, L.M. / Merrihew, R.V. / Huet, S. / Willson, T.M. |
External links | Bioorg. Med. Chem. Lett. / PubMed:18722772 |
Methods | X-ray diffraction |
Resolution | 2.9 Å |
Structure data | PDB-3dy6: |
Chemicals | ChemComp-IOD: ChemComp-DY6: ChemComp-HOH: |
Source |
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Keywords | TRANSCRIPTION / PPAR / nulear receptor / Activator / DNA-binding / Metal-binding / Nucleus / Transcription regulation / Zinc-finger |