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TitleDiscovery and Initial SAR of Arylsulfonylpiperazine Inhibitors of 11beta-Hydroxysteroid Dehydrogenase Type 1 (11beta-HSD1)
Journal, issue, pagesBioorg. Med. Chem. Lett., Vol. 18, Page 3513-3516, Year 2008
Publish dateApr 29, 2008 (structure data deposition date)
AuthorsSun, D. / Wang, Z. / Di, Y. / Jaen, J.C. / Labelle, M. / Ma, J. / Miao, S. / Sudom, A. / Tang, L. / Tomooka, C.S. ...Sun, D. / Wang, Z. / Di, Y. / Jaen, J.C. / Labelle, M. / Ma, J. / Miao, S. / Sudom, A. / Tang, L. / Tomooka, C.S. / Tu, H. / Ursu, S. / Walker, N. / Yan, X. / Ye, Q. / Powers, J.P.
External linksBioorg. Med. Chem. Lett. / PubMed:18511278
MethodsX-ray diffraction
Resolution2.35 Å
Structure data

PDB-3czr:
Crystal Structure of Human 11-beta-Hydroxysteroid Dehydrogenase (HSD1) in Complex with Arylsulfonylpiperazine Inhibitor
Method: X-RAY DIFFRACTION / Resolution: 2.35 Å

Chemicals

ChemComp-NAP:
NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE

ChemComp-3CZ:
(2R)-1-[(4-tert-butylphenyl)sulfonyl]-2-methyl-4-(4-nitrophenyl)piperazine

ChemComp-CPS:
3-[(3-CHOLAMIDOPROPYL)DIMETHYLAMMONIO]-1-PROPANESULFONATE / detergent*YM

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsOXIDOREDUCTASE / 11beta / hydroxysteroid / dehydrogenase / Endoplasmic reticulum / Glycoprotein / Lipid metabolism / Membrane / Microsome / NADP / Polymorphism / Signal-anchor / Steroid metabolism / Transmembrane

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