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-Structure paper
Title | Antitumor activity and pharmacology of a selective focal adhesion kinase inhibitor, PF-562,271. |
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Journal, issue, pages | Cancer Res., Vol. 68, Page 1935-1944, Year 2008 |
Publish date | Jan 17, 2008 (structure data deposition date) |
![]() | Roberts, W.G. / Ung, E. / Whalen, P. / Cooper, B. / Hulford, C. / Autry, C. / Richter, D. / Emerson, E. / Lin, J. / Kath, J. ...Roberts, W.G. / Ung, E. / Whalen, P. / Cooper, B. / Hulford, C. / Autry, C. / Richter, D. / Emerson, E. / Lin, J. / Kath, J. / Coleman, K. / Yao, L. / Martinez-Alsina, L. / Lorenzen, M. / Berliner, M. / Luzzio, M. / Patel, N. / Schmitt, E. / LaGreca, S. / Jani, J. / Wessel, M. / Marr, E. / Griffor, M. / Vajdos, F. |
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Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | ![]() PDB-3bz3: |
Chemicals | ![]() ChemComp-YAM: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / kinase / DFG-helix / Acetylation / Alternative splicing / ATP-binding / Cell junction / Nucleotide-binding / Phosphoprotein / Tyrosine-protein kinase |