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-Structure paper
Title | Tyramine fragment binding to BACE-1 |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 18, Page 1304-1307, Year 2008 |
Publish date | Dec 21, 2007 (structure data deposition date) |
![]() | Kuglstatter, A. / Stahl, M. / Peters, J.U. / Huber, W. / Stihle, M. / Schlatter, D. / Benz, J. / Ruf, A. / Roth, D. / Enderle, T. / Hennig, M. |
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Methods | X-ray diffraction |
Resolution | 2.3 - 2.5 Å |
Structure data | ![]() PDB-3bra: ![]() PDB-3buf: ![]() PDB-3bug: ![]() PDB-3buh: |
Chemicals | ![]() ChemComp-AEF: ![]() ChemComp-HOH: ![]() ChemComp-AEG: ![]() ChemComp-AEH: ![]() ChemComp-AED: |
Source |
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![]() | HYDROLASE / ALZHEIMER'S DISEASE / ASPARTIC PROTEASE / BETA-SECRETASE / MEMAPSIN 2 / FRAGMENT SCREEN / Alternative splicing / Aspartyl protease / Glycoprotein / Membrane / Transmembrane / Zymogen |