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-Structure paper
Title | Bace-1 Inhibitors Part 3: Identification of Hydroxy Ethylamines (Heas) with Nanomolar Potency in Cells. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 18, Page 1022-, Year 2008 |
Publish date | Dec 4, 2007 (structure data deposition date) |
![]() | Beswick, P. / Charrier, N. / Clarke, B. / Demont, E. / Dingwall, C. / Dunsdon, R. / Faller, A. / Gleave, R. / Hawkins, J. / Hussain, I. ...Beswick, P. / Charrier, N. / Clarke, B. / Demont, E. / Dingwall, C. / Dunsdon, R. / Faller, A. / Gleave, R. / Hawkins, J. / Hussain, I. / Johnson, C.N. / Macpherson, D. / Maile, G. / Matico, R. / Milner, P. / Mosley, J. / Naylor, A. / O'Brien, A. / Redshaw, S. / Riddell, D. / Rowland, P. / Skidmore, J. / Soleil, V. / Smith, K.J. / Stanway, S. / Stemp, G. / Stuart, A. / Sweitzer, S. / Theobald, P. / Vesey, D. / Walter, D.S. / Ward, J. / Wayne, G. |
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Methods | X-ray diffraction |
Resolution | 1.6 Å |
Structure data | ![]() PDB-2vij: |
Chemicals | ![]() ChemComp-C44: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE / ALTERNATIVE SPLICING / BETA-SITE APP CLEAVING ENZYME / BETA-SECRETASE / ASPARTYL PROTEASE / ASP-2 / BACE-1 / ZYMOGEN / PROTEASE / MEMBRANE / MEMAPSIN-2 / GLYCOPROTEIN / TRANSMEMBRANE |