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Title7-fluoroindazoles as potent and selective inhibitors of factor xa.
Journal, issue, pagesJ. Med. Chem., Vol. 51, Page 282-297, Year 2008
Publish dateSep 14, 2007 (structure data deposition date)
AuthorsLee, Y.K. / Parks, D.J. / Lu, T. / Thieu, T.V. / Markotan, T. / Pan, W. / McComsey, D.F. / Milkiewicz, K.L. / Crysler, C.S. / Ninan, N. ...Lee, Y.K. / Parks, D.J. / Lu, T. / Thieu, T.V. / Markotan, T. / Pan, W. / McComsey, D.F. / Milkiewicz, K.L. / Crysler, C.S. / Ninan, N. / Abad, M.C. / Giardino, E.C. / Maryanoff, B.E. / Damiano, B.P. / Player, M.R.
External linksJ. Med. Chem. / PubMed:18159923
MethodsX-ray diffraction
Resolution2.3 Å
Structure data

PDB-2ra0:
X-ray Structure of FXa in complex with 7-fluoroindazole
Method: X-RAY DIFFRACTION / Resolution: 2.3 Å

Chemicals

ChemComp-JNJ:
1-(3-amino-1,2-benzisoxazol-5-yl)-6-(4-{2-[(dimethylamino)methyl]-1H-imidazol-1-yl}-2-fluorophenyl)-7-fluoro-1H-indazole-3-carboxamide

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsHYDROLASE / serine protease / Blood coagulation / Calcium / Cleavage on pair of basic residues / EGF-like domain / Gamma-carboxyglutamic acid / Glycoprotein / Hydroxylation / Polymorphism / Zymogen

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