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| Title | Molecular analysis of the HIV-1 resistance development: enzymatic activities, crystal structures, and thermodynamics of nelfinavir-resistant HIV protease mutants |
|---|---|
| Journal, issue, pages | J. Mol. Biol., Vol. 374, Page 1005-1016, Year 2007 |
| Publish date | May 16, 2007 (structure data deposition date) |
Authors | Kozisek, M. / Bray, J. / Rezacova, P. / Saskova, K. / Brynda, J. / Pokorna, J. / Mammano, F. / Rulisek, L. / Konvalinka, J. |
External links | J. Mol. Biol. / PubMed:17977555 |
| Methods | X-ray diffraction |
| Resolution | 1.85 - 2.5 Å |
| Structure data | ![]() PDB-2pym: ![]() PDB-2pyn: ![]() PDB-2q63: ![]() PDB-2q64: |
| Chemicals | ![]() ChemComp-1UN: ![]() ChemComp-HOH: |
| Source |
|
Keywords | HYDROLASE / resistance; nelfinavir |
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human immunodeficiency virus 1
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