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-Structure paper
Title | Inhibition of Monometalated Methionine Aminopeptidase: Inhibitor Discovery and Crystallographic Analysis. |
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Journal, issue, pages | J. Med. Chem., Vol. 50, Page 5735-5742, Year 2007 |
Publish date | Mar 24, 2007 (structure data deposition date) |
Authors | Huang, M. / Xie, S.X. / Ma, Z.Q. / Huang, Q.Q. / Nan, F.J. / Ye, Q.Z. |
External links | J. Med. Chem. / PubMed:17948983 |
Methods | X-ray diffraction |
Resolution | 1.6 - 1.8 Å |
Structure data | PDB-2p98: PDB-2p99: PDB-2p9a: |
Chemicals | ChemComp-MN: ChemComp-NA: ChemComp-YE7: ChemComp-HOH: ChemComp-YE6: |
Source |
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Keywords | HYDROLASE / monometalated / mononuclear / Mn(II)-form / enzyme-inhibitor complex / metalloenzyme / dimetalated / dinuclear |