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-Structure paper
Title | Crystal Structure of the T315I Abl Mutant in Complex with the Aurora Kinases Inhibitor Pha-739358. |
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Journal, issue, pages | Cancer Res., Vol. 67, Page 7987-, Year 2007 |
Publish date | Jul 27, 2007 (structure data deposition date) |
Authors | Modugno, M. / Casale, E. / Soncini, C. / Rosettani, P. / Colombo, R. / Lupi, R. / Rusconi, L. / Fancelli, D. / Carpinelli, P. / Cameron, A.D. ...Modugno, M. / Casale, E. / Soncini, C. / Rosettani, P. / Colombo, R. / Lupi, R. / Rusconi, L. / Fancelli, D. / Carpinelli, P. / Cameron, A.D. / Isacchi, A. / Moll, J. |
External links | Cancer Res. / PubMed:17804707 |
Methods | X-ray diffraction |
Resolution | 2.5 Å |
Structure data | PDB-2v7a: |
Chemicals | ChemComp-627: ChemComp-MG: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / KINASE / NUCLEUS / MYRISTATE / CYTOPLASM / MANGANESE / CELL ADHESION / METAL-BINDING / PROTO-ONCOGENE / TYROSINE-PROTEIN KINASE / CHROMOSOMAL REARRANGEMENT / LIPOPROTEIN / POLYMORPHISM / CYTOSKELETON / MAGNESIUM / SH2 DOMAIN / SH3 DOMAIN / ATP-BINDING / NUCLEOTIDE-BINDING / ALTERNATIVE SPLICING / PHOSPHORYLATION / KINASE INHIBITOR / T315I ABL MUTANT |