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-Structure paper
Title | Compensating enthalpic and entropic changes hinder binding affinity optimization. |
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Journal, issue, pages | Chem. Biol. Drug Des., Vol. 69, Page 413-422, Year 2007 |
Publish date | Apr 17, 2007 (structure data deposition date) |
![]() | Lafont, V. / Armstrong, A.A. / Ohtaka, H. / Kiso, Y. / Mario Amzel, L. / Freire, E. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.45 - 1.9 Å |
Structure data | ![]() PDB-2pk5: ![]() PDB-2pk6: |
Chemicals | ![]() ChemComp-075: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-O33: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / PROTEASE COMPLEX / Viral Protein / HYDROLASE-HYDROLASE INHIBITOR complex |