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-Structure paper
Title | Indolinone based phosphoinositide-dependent kinase-1 (PDK1) inhibitors. Part 2: Optimization of BX-517. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 17, Page 3819-3825, Year 2007 |
Publish date | Apr 1, 2007 (structure data deposition date) |
![]() | Islam, I. / Brown, G. / Bryant, J. / Hrvatin, P. / Kochanny, M.J. / Phillips, G.B. / Yuan, S. / Adler, M. / Whitlow, M. / Lentz, D. ...Islam, I. / Brown, G. / Bryant, J. / Hrvatin, P. / Kochanny, M.J. / Phillips, G.B. / Yuan, S. / Adler, M. / Whitlow, M. / Lentz, D. / Polokoff, M.A. / Wu, J. / Shen, J. / Walters, J. / Ho, E. / Subramanyam, B. / Zhu, D. / Feldman, R.I. / Arnaiz, D.O. |
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Methods | X-ray diffraction |
Resolution | 2.13 Å |
Structure data | ![]() PDB-2pe2: |
Chemicals | ![]() ChemComp-SO4: ![]() ChemComp-464: ![]() ChemComp-GOL: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / PROTEIN INHIBITOR COMPLEX / SERINE KINASE |