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-Structure paper
Title | Discovery of non-covalent dipeptidyl peptidase IV inhibitors which induce a conformational change in the active site. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 17, Page 1765-1768, Year 2007 |
Publish date | Jan 9, 2007 (structure data deposition date) |
![]() | Sheehan, S.M. / Mest, H.J. / Watson, B.M. / Klimkowski, V.J. / Timm, D.E. / Cauvin, A. / Parsons, S.H. / Shi, Q. / Canada, E.J. / Wiley, M.R. ...Sheehan, S.M. / Mest, H.J. / Watson, B.M. / Klimkowski, V.J. / Timm, D.E. / Cauvin, A. / Parsons, S.H. / Shi, Q. / Canada, E.J. / Wiley, M.R. / Ruehter, G. / Evers, B. / Petersen, S. / Blaszczak, L.C. / Pulley, S.R. / Margolis, B.J. / Wishart, G.N. / Renson, B. / Hankotius, D. / Mohr, M. / Zechel, J.C. / Michael Kalbfleisch, J. / Dingess-Hammond, E.A. / Boelke, A. / Weichert, A.G. |
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Methods | X-ray diffraction |
Resolution | 2.1 Å |
Structure data | ![]() PDB-2ogz: |
Chemicals | ![]() ChemComp-U1N: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE / DIPEPTIDYL PEPTIDASE IV / CD26 / DPIV / DPP-IV / DPP4 / Serine Protease / inhibitor |