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-Structure paper
Title | Structural and Mechanistic Studies on the Inhibition of the Hypoxia-Inducible Transcription Factor Hydroxylases by Tricarboxylic Acid Cycle Intermediates. |
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Journal, issue, pages | J. Biol. Chem., Vol. 282, Page 3293-3301, Year 2007 |
Publish date | Mar 9, 2006 (structure data deposition date) |
![]() | Hewitson, K. / Lienard, B. / McDonough, M.A. / Clifton, I.J. / Butler, D. / Soares, A.S. / Oldham, N.J. / McNeill, L.A. / Schofield, C.J. |
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Methods | X-ray diffraction |
Resolution | 2.3 - 2.4 Å |
Structure data | ![]() PDB-2cgn: ![]() PDB-2cgo: |
Chemicals | ![]() ChemComp-FE: ![]() ChemComp-SIN: ![]() ChemComp-SO4: ![]() ChemComp-HOH: ![]() ChemComp-FUM: |
Source |
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![]() | OXIDOREDUCTASE / 2-OXOGLUTARATE / ACETYLATION / ACTIVATOR / ALTERNATIVE SPLICING / ASPARAGINYL HYDROXYLASE / DNA-BINDING / DSBH / FI / HIF / HYDROXYLATION / HYPOXIA / NUCLEAR PROTEIN / OXYGENASE / PHOSPHORYLATION / POLYMORPHISM / S-NITROSYLATION / TRANSCRIPTION / TRANSCRIPTION ACTIVATOR/INHIBITOR / TRANSCRIPTION REGULATION / DIOXYGENASE / IRON / METAL-BINDING |