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-Structure paper
Title | Design of potent inhibitors of human beta-secretase. Part 2. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 17, Page 78-81, Year 2007 |
Publish date | Jul 10, 2006 (structure data deposition date) |
![]() | Freskos, J.N. / Fobian, Y.M. / Benson, T.E. / Moon, J.B. / Bienkowski, M.J. / Brown, D.L. / Emmons, T.L. / Heintz, R. / Laborde, A. / McDonald, J.J. ...Freskos, J.N. / Fobian, Y.M. / Benson, T.E. / Moon, J.B. / Bienkowski, M.J. / Brown, D.L. / Emmons, T.L. / Heintz, R. / Laborde, A. / McDonald, J.J. / Mischke, B.V. / Molyneaux, J.M. / Mullins, P.B. / Bryan Prince, D. / Paddock, D.J. / Tomasselli, A.G. / Winterrowd, G. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | ![]() PDB-2hm1: |
Chemicals | ![]() ChemComp-LIQ: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE / protein-inhibitor complex |