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-Structure paper
Title | Crystal structure of the Mycobacterium tuberculosis P450 CYP121-fluconazole complex reveals new azole drug-P450 binding mode. |
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Journal, issue, pages | J. Biol. Chem., Vol. 281, Page 39437-39443, Year 2006 |
Publish date | Sep 29, 2006 (structure data deposition date) |
![]() | Seward, H.E. / Roujeinikova, A. / McLean, K.J. / Munro, A.W. / Leys, D. |
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Methods | X-ray diffraction |
Resolution | 1.6 - 1.9 Å |
Structure data | ![]() PDB-2ij5: ![]() PDB-2ij7: |
Chemicals | ![]() ChemComp-SO4: ![]() ChemComp-HEM: ![]() ChemComp-HOH: ![]() ChemComp-TPF: |
Source |
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![]() | OXIDOREDUCTASE / tuberculosis / CYP121 / cytochrome P450 / azole ligation / fluconazole / P450 CYP121 / azole drug |