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-Structure paper
Title | Structural basis of Src tyrosine kinase inhibition with a new class of potent and selective trisubstituted purine-based compounds. |
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Journal, issue, pages | Chem. Biol. Drug Des., Vol. 67, Page 46-57, Year 2006 |
Publish date | Oct 20, 2005 (structure data deposition date) |
![]() | Dalgarno, D. / Stehle, T. / Narula, S. / Schelling, P. / van Schravendijk, M.R. / Adams, S. / Andrade, L. / Keats, J. / Ram, M. / Jin, L. ...Dalgarno, D. / Stehle, T. / Narula, S. / Schelling, P. / van Schravendijk, M.R. / Adams, S. / Andrade, L. / Keats, J. / Ram, M. / Jin, L. / Grossman, T. / MacNeil, I. / Metcalf III, C. / Shakespeare, W. / Wang, Y. / Keenan, T. / Sundaramoorthi, R. / Bohacek, R. / Weigele, M. / Sawyer, T. |
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Methods | X-ray diffraction |
Resolution | 2.1 - 2.5 Å |
Structure data | ![]() PDB-2bdf: ![]() PDB-2bdj: |
Chemicals | ![]() ChemComp-24A: ![]() ChemComp-HOH: ![]() ChemComp-HET: |
Source |
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![]() | TRANSFERASE / Src Kinase Inhibitor |