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-Structure paper
Title | Synthesis and evaluation of arylaminoethyl amides as noncovalent inhibitors of cathepsin S. Part 3: Heterocyclic P3. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 16, Page 1975-1980, Year 2006 |
Publish date | Nov 14, 2005 (structure data deposition date) |
Authors | Tully, D.C. / Liu, H. / Alper, P.B. / Chatterjee, A.K. / Epple, R. / Roberts, M.J. / Williams, J.A. / Nguyen, K.T. / Woodmansee, D.H. / Tumanut, C. ...Tully, D.C. / Liu, H. / Alper, P.B. / Chatterjee, A.K. / Epple, R. / Roberts, M.J. / Williams, J.A. / Nguyen, K.T. / Woodmansee, D.H. / Tumanut, C. / Li, J. / Spraggon, G. / Chang, J. / Tuntland, T. / Harris, J.L. / Karanewsky, D.S. |
External links | Bioorg. Med. Chem. Lett. / PubMed:16446091 |
Methods | X-ray diffraction |
Resolution | 1.9 Å |
Structure data | PDB-2f1g: |
Chemicals | ChemComp-GNF: ChemComp-GOL: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / Cathepsin S / noncovalent / inhibition / 2-(Benzooxazol-2-ylamino) acetamides |