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-Structure paper
Title | Structure-Based Design of Protein Tyrosine Phosphatase-1B Inhibitors |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 15, Page 2503-, Year 2005 |
Publish date | Dec 21, 2004 (structure data deposition date) |
Authors | Black, E. / Breed, J. / Breeze, A.L. / Embrey, K. / Garcia, R. / Gero, T.W. / Godfrey, L. / Kenny, P.W. / Morley, A.D. / Minshull, C.A. ...Black, E. / Breed, J. / Breeze, A.L. / Embrey, K. / Garcia, R. / Gero, T.W. / Godfrey, L. / Kenny, P.W. / Morley, A.D. / Minshull, C.A. / Pannifer, A.D. / Read, J. / Rees, A. / Russell, D.J. / Toader, D. / Tucker, J. |
External links | Bioorg. Med. Chem. Lett. / PubMed:15863305 |
Methods | X-ray diffraction |
Resolution | 1.8 - 2.4 Å |
Structure data | PDB-2bgd: PDB-2bge: |
Chemicals | ChemComp-T1D: ChemComp-CL: ChemComp-PO4: ChemComp-NA: ChemComp-HOH: ChemComp-T2D: |
Source |
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Keywords | HYDROLASE / PROTEIN TYROSINE PHOSPHATASE / 1 / 2 / 5-THIADIAZOLIDIN-3-ONE-1 / 1-DIOXIDE TEMPLATE |