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-Structure paper
Title | Role of hydroxyl group and R/S configuration of isostere in binding properties of HIV-1 protease inhibitors |
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Journal, issue, pages | Eur. J. Biochem., Vol. 271, Page 4451-4461, Year 2004 |
Publish date | Jun 12, 2002 (structure data deposition date) |
![]() | Petrokova, H. / Duskova, J. / Dohnalek, J. / Skalova, T. / Vondrackova-Buchtelova, E. / Soucek, M. / Konvalinka, J. / Brynda, J. / Fabry, M. / Sedlacek, J. / Hasek, J. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.45 Å |
Structure data | ![]() PDB-1m0b: |
Chemicals | ![]() ChemComp-0ZQ: ![]() ChemComp-GOL: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / HIV PROTEASE / PEPTIDOMIMETICS / HYDROLASE-HYDROLASE INHIBITOR complex |