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-Structure paper
Title | SAR and factor IXa crystal structure of a dual inhibitor of factors IXa and Xa |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 14, Page 5263-5267, Year 2004 |
Publish date | Aug 13, 2004 (structure data deposition date) |
![]() | Smallheer, J.M. / Alexander, R.S. / Wang, J. / Wang, S. / Nakajima, S. / Rossi, K.A. / Smallwood, A. / Barbera, F. / Burdick, D. / Luettgen, J.M. ...Smallheer, J.M. / Alexander, R.S. / Wang, J. / Wang, S. / Nakajima, S. / Rossi, K.A. / Smallwood, A. / Barbera, F. / Burdick, D. / Luettgen, J.M. / Knabb, R.M. / Wexler, R.R. / Jadhav, P.K. |
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Methods | X-ray diffraction |
Resolution | 2.9 Å |
Structure data | ![]() PDB-1x7a: |
Chemicals | ![]() ChemComp-187: |
Source |
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![]() | blood clotting / hydrolase / inhibition; X-ray structure |