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-Structure paper
Title | The protein kinase C inhibitor bisindolyl maleimide 2 binds with reversed orientations to different conformations of protein kinase a. |
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Journal, issue, pages | J. Biol. Chem., Vol. 279, Page 23679-23690, Year 2004 |
Publish date | Apr 6, 2004 (structure data deposition date) |
Authors | Gassel, M. / Breitenlechner, C.B. / Koenig, N. / Huber, R. / Engh, R.A. / Bossemeyer, D. |
External links | J. Biol. Chem. / PubMed:14996846 |
Methods | X-ray diffraction |
Resolution | 2.5 Å |
Structure data | PDB-1szm: |
Chemicals | ChemComp-BI4: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / PKA / PKC / bisindolyl maleimide 2 / LY333531 / selectivity / surrogate kinase / amino acid residue exchange |