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Title | DESIGN OF WEAKLY BASIC THROMBIN INHIBITORS INCORPORATING NOVEL P1 BINDING FUNCTIONS: MOLECULAR AND X-RAY CRYSTALLOGRAPHIC STUDIES |
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Journal, issue, pages | Biochemistry, Vol. 42, Page 9013-9021, Year 2003 |
Publish date | Jan 16, 2003 (structure data deposition date) |
![]() | De Simone, G. / Menchise, V. / Omaggio, S. / Pedone, C. / Scozzafava, A. / Supuran, C.T. |
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Methods | X-ray diffraction |
Resolution | 1.9 Å |
Structure data | ![]() PDB-1no9: |
Chemicals | ![]() ChemComp-NAG: ![]() ChemComp-4ND: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / COMPLEX (SERINE PROTEASE-INHIBITOR) / BLOOD COAGULATION / SERINE PROTEINASE INHIBITION / N / N-DIPHENYLCARBAMOYL-AMINOGUANIDINE / HYDROLASE / HYDROLASE-HYDROLASE INHIBITOR COMPLEX |