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-Structure paper
Title | Discovery of a Novel Series of 6-Azauracil-Based Thyroid Hormone Receptor Ligands: Potent, TRbeta Subtype-Selective Thyromimetics |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 13, Page 379-382, Year 2003 |
Publish date | Oct 30, 2002 (structure data deposition date) |
Authors | Dow, R.L. / Schneider, S.R. / Paight, E.S. / Hank, R.F. / Chiang, P. / Cornelius, P. / Lee, E. / Newsome, W.P. / Swick, A.G. / Spitzer, J. ...Dow, R.L. / Schneider, S.R. / Paight, E.S. / Hank, R.F. / Chiang, P. / Cornelius, P. / Lee, E. / Newsome, W.P. / Swick, A.G. / Spitzer, J. / Hargrove, D.M. / Patterson, T.A. / Pandit, J. / Chrunyk, B.A. / LeMotte, P.K. / Danley, D.E. / Rosner, M.H. / Ammirati, M.J. / Simons, S.P. / Schulte, G.K. / Tate, B.F. / DaSilva-Jardine, P. |
External links | Bioorg. Med. Chem. Lett. / PubMed:12565933 |
Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | PDB-1n46: |
Chemicals | ChemComp-PFA: ChemComp-HOH: |
Source |
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Keywords | TRANSCRIPTION |