eF-site ID 4p6w-AB
PDB Code 4p6w
Chain A, B

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Title Crystal Structure of mometasone furoate-bound glucocorticoid receptor ligand binding domain
Classification HORMONE RECEPTOR/HORMONE ACTIVATOR
Compound Glucocorticoid receptor
Source (NCOA2_HUMAN)
Sequence A:  PQLTPTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNM
LGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMALMA
FALGWRSYRQSSANLLYFAPDLIINEQRMTLPCMYDQCKH
MLYVSSELHRLQVSYEEYLCMKVLLLLSTIPKDGLKSQEL
FDEIRMTYIKELGAAIVAREGNSSQNWQRFYQLTKLLDSM
HEVVENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYS
NGNIKKLLFHQK
B:  ANALLRYLLDKD
Description


Functional site

1) chain A
residue 560
type
sequence M
description binding site for residue MOF A 801
source : AC1

2) chain A
residue 563
type
sequence L
description binding site for residue MOF A 801
source : AC1

3) chain A
residue 564
type
sequence N
description binding site for residue MOF A 801
source : AC1

4) chain A
residue 567
type
sequence G
description binding site for residue MOF A 801
source : AC1

5) chain A
residue 570
type
sequence Q
description binding site for residue MOF A 801
source : AC1

6) chain A
residue 600
type
sequence W
description binding site for residue MOF A 801
source : AC1

7) chain A
residue 601
type
sequence M
description binding site for residue MOF A 801
source : AC1

8) chain A
residue 604
type
sequence M
description binding site for residue MOF A 801
source : AC1

9) chain A
residue 611
type
sequence R
description binding site for residue MOF A 801
source : AC1

10) chain A
residue 623
type
sequence F
description binding site for residue MOF A 801
source : AC1

11) chain A
residue 639
type
sequence M
description binding site for residue MOF A 801
source : AC1

12) chain A
residue 642
type
sequence Q
description binding site for residue MOF A 801
source : AC1

13) chain A
residue 646
type
sequence M
description binding site for residue MOF A 801
source : AC1

14) chain A
residue 735
type
sequence Y
description binding site for residue MOF A 801
source : AC1

15) chain A
residue 736
type
sequence C
description binding site for residue MOF A 801
source : AC1

16) chain A
residue 739
type
sequence T
description binding site for residue MOF A 801
source : AC1

17) chain A
residue 749
type
sequence F
description binding site for residue MOF A 801
source : AC1

18) chain A
residue 703
type CROSSLNK
sequence A
description Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO) => ECO:0000269|PubMed:12144530
source Swiss-Prot : SWS_FT_FI1


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