eF-site ID 2w8y-A
PDB Code 2w8y
Chain A

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Title RU486 bound to the progesterone receptor in a destabilized agonistic conformation
Classification RECEPTOR
Compound PROGESTERONE RECEPTOR
Source Homo sapiens (Human) (PRGR_HUMAN)
Sequence A:  LIPPLINLLMSIEPDVIYAGHDNTKPDTSSSLLTSLNQLG
ERQLLSVVKWSKSLPGFRNLHIDDQITLIQYSWMSLMVFG
LGWRSYKHVSGQMLYFAPDLILNEQRMKESSFYSLCLTMW
QIPQEFVKLQVSQEEFLCMKVLLLLNTIPLEGLRSQTQFE
EMRSSYIRELIKAIGLRQKGVVSSSQRFYQLTKLLDNLHD
LVKQLHLYCLNTFIQSRALSVEFPEMMSEVIAAQLPKILA
GMVKPLLFHKK
Description


Functional site

1) chain A
residue 715
type
sequence L
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

2) chain A
residue 718
type
sequence L
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

3) chain A
residue 719
type
sequence N
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

4) chain A
residue 721
type
sequence L
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

5) chain A
residue 722
type
sequence G
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

6) chain A
residue 723
type
sequence E
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

7) chain A
residue 725
type
sequence Q
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

8) chain A
residue 755
type
sequence W
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

9) chain A
residue 756
type
sequence M
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

10) chain A
residue 759
type
sequence M
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

11) chain A
residue 766
type
sequence R
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

12) chain A
residue 794
type
sequence F
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

13) chain A
residue 797
type
sequence L
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

14) chain A
residue 801
type
sequence M
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

15) chain A
residue 890
type
sequence Y
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

16) chain A
residue 891
type
sequence C
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

17) chain A
residue 909
type
sequence M
description BINDING SITE FOR RESIDUE 486 A 1000
source : AC1

18) chain A
residue 737
type
sequence P
description BINDING SITE FOR RESIDUE SO4 A 1934
source : AC4

19) chain A
residue 738
type
sequence G
description BINDING SITE FOR RESIDUE SO4 A 1934
source : AC4

20) chain A
residue 740
type
sequence R
description BINDING SITE FOR RESIDUE SO4 A 1934
source : AC4

21) chain A
residue 741
type
sequence N
description BINDING SITE FOR RESIDUE SO4 A 1934
source : AC4

22) chain A
residue 766
type BINDING
sequence R
description BINDING => ECO:0000269|PubMed:9620806
source Swiss-Prot : SWS_FT_FI1


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